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CAS Name (Chinese) Name (English) Application
1094322-91-4 霉酚酸酯B 1-[2-(4-Morpholinyl)ethoxy] Prevention and treatment of kidney, liver, and heart transplant rejection.
619-100-6 吉西他滨 Gemcitabine Antineoplastic drugs
79902-63-9 辛伐他汀 Simvastatin Reduces cholesterol, LDL (low-density lipoprotein), and VLDL (very-low-density lipoprotein) cholesterol.
486460-32-6 西他列汀 Sitagliptin Inhibitor drugs for the treatment of type 2 diabetes.
127852-28-2 福沙匹坦 (R)-1-[3,5-Bis(trifluoromethyl)phenyl]ethanol Prevention of chemotherapy-induced nausea and vomiting (CINV).
59729-33-8 西酞普兰 Citalopram Antidepressant medications
850649-61-5 阿格列汀 ALOGLIPTIN(ALOGLIPTINE, ALOGLIPTINA) Antihyperglycemic agents
144689-24-7 奥美沙坦 Olmesartan Antihypertensive drugs
144689-78-1 奥美沙坦酯 Olmesartan Antihypertensive drugs
120014-06-4 多奈哌齐 Donepezil Alzheimer disease
103628-46-2 舒马曲坦 Sumatriptan Migraine (w/ or w/o aura);Dural inflamm
202138-50-9 泰诺福韦酯 Tenofovir disoproxil fumarate Antiviral agent; indicated for HIV and chronic HBV infection.
303-53-7 环苯扎林 CYCLOBENZAPRINE HCL Relief of pain and discomfort associated with muscle spasms.
82410-32-0 更昔洛韦 Ganciclovir CMV infection (immunocompromised); CMV retinitis maintenance (AIDS)
130018-77-8 左西替利嗪 Levocetirizine Antiallergic drug that works by blocking histamine in allergic reactions.
90357-06-5 比卡鲁胺 Bicalutamide Prostate cancer
18323-44-9 克林霉素 Clindamycin Treatment of common infections caused by susceptible bacteria.
1951-25-3 胺碘酮 Amiodarone Class Ⅲ antiarrhythmic drugs
97832-05-8 苯达莫司汀 Bendamustine Alkylating agent; primarily for hematologic malignancies including CLL and NHL.
74578-69-1 头孢曲松钠 Ceftriaxone sodium Third-generation cephalosporin antibiotics
81110-73-8 卡多曲 Racecadotril Relief of acute diarrhea symptoms
183198-49-4 地氯雷他定 Desloratadine Second-generation antihistamine for allergy relief
39809-25-1 喷昔洛韦 Penciclovir Severe forms of shingles
19794-93-5 曲唑酮 Trazodone Depression, particularly in elderly patients or those with cardiac conditions.
86386-73-4 氟康唑 Fluconazole Systemic candidiasis
668270-12-0 利格列汀 Linagliptin For adult patients with type 2 diabetes
106266-06-2 利培酮 Risperidone For adolescents (13 years and older) and adults with schizophrenia
82248-59-7 阿托莫西汀 Atomoxetine hydrochloride Non-CNS stimulant drugs for ADHD
1009119-64-5 达卡他韦 Daclatasvir Direct-acting antiviral (DAA) for chronic hepatitis C virus (HCV) infection.
73590-58-6 奥美拉唑 Omeprazole For duodenal ulcers and Zollinger-Ellison syndrome; also for gastric ulcers and reflux esophagitis.
88040-23-7 头孢吡肟 Cefepime Fourth-generation cephalosporin; for respiratory, urinary, skin/soft tissue, and intra-abdominal infections.
147098-20-2 瑞舒伐他汀钙 Rosuvastatin calcium Primary hypercholesterolemia (IIa, incl. HeFH) / mixed dyslipidemia (IIb); uncontrolled by diet/exercise.
274901-16-5 维达列汀 Vildagliptin DPP-4 inhibitor; T2DM glycemic control
32222-06-3 骨化三醇 Calcitriol Osteoporosis in older adults
459789-99-2 奥贝胆酸 Obeticholic Acid Bile acid analog; PBC; NASH-related liver disease
104227-87-4 泛昔洛韦 Famciclovir Shingles and primary genital herpes
171596-29-5 他达那非 Tadalafil Treatment of erectile dysfunction (ED) and pulmonary arterial hypertension (PAH).
120092-68-4 马尼地平 Manidipine Antihypertensive drugs
100427-26-7 乐卡地平 Lercanidipine DHP-CCB (new-gen); mild-moderate hypertension
59-05-2 甲氨蝶呤 Methotrexate Antifolate; cancer/RA; DHFR inhibitor
13189-98-5 福多司坦 Fudosteine Thick sputum; respiratory conditions
128-62-1 那可汀 Narcotine Bronchial antispasmodic antitussives
50-33-9 保泰松 Phenylbutazone NSAID for rheumatic arthritis, rheumatoid arthritis, and acute gout.
99592-32-2 舍他康唑 Sertaconazole nitrate Broad-spectrum antifungal; cutaneous/mucosal infections
18559-94-9 沙丁胺醇 Salbutamol SABA; inhibits histamine release; prevents bronchospasm
55981-09-4 硝唑尼特 Nitazoxanide Broad-spectrum antiparasitic: Cryptosporidium/Giardia; + antiviral/antibacterial
173903-47-4 替唑尼特 TIZOXANIDE Nitroimidazole: anaerobes; Giardia/Entamoeba
143491-57-0 恩曲他滨 Emtricitabine Treatment of HIV-1 infection in adults
134678-17-4 拉米夫定 Lamivudine Treatment of HIV-1 infection
107667-60-7 聚普瑞锌 Polaprezinc Gastric protectant; gastric ulcer adjunct
241479-67-4 艾莎康唑 Isavuconazole Triazole antifungal: invasive aspergillosis/mucormycosis (adults)
171228-49-2 泊沙康唑 Posaconazole Enteric tablets/suspension: prevent invasive Aspergillus/Candida in immunocompromised patients ≥13 yrs at high risk.
864821-90-9 伊卢多啉 Eluxadoline μ/κ agonist & δ antagonist; IBS-D
74682-62-5 替卡西林钠 Ticarcillin sodium Broad-spectrum penicillin: Gram-negative bacteria (e.g., P. aeruginosa, E. coli)
81110-73-8 消旋卡多曲 Racecadotril Acute diarrhea: adults (watery); infants/children >1 mo; traveler's diarrhea
89786-04-9 他唑巴坦 Tazobactam acid β-lactamase inhibitor + β-lactam (e.g., piperacillin); enhances activity vs. MDROs; serious infections
99592-32-2 舍他康唑 Sertaconazole nitrate Broad-spectrum antifungal; cutaneous/mucosal infections
65576-45-6 阿塞那平 Asenapine Antipsychotic: schizophrenia; bipolar mania
21679-14-1 氟达拉滨 Fludarabine Antineoplastic drugs
154361-50-9 卡培他滨 Capecitabine Antineoplastic: adjuvant colon cancer (Dukes' C, post-resection, fluoropyrimidine monotherapy); adjuvant intrahepatic cholangiocarcinoma (post-op)
486460-32-6 磷酸西他列汀 Sitagliptin Oral DPP-4 inhibitor; T2DM glycemic control
151096-09-2 莫西沙星 Moxifloxacin Acute bacterial sinusitis: S. pneumoniae, H. influenzae, M. catarrhalis
112811-59-3 加替沙星 Gatifloxacin Gatifloxacin: 4th-gen fluoroquinolone; broad-spectrum (Gram+/Gram-); most potent vs. Gram-
119141-88-7 埃索美拉唑 Esomeprazole PPI: GERD, gastric ulcer, acid-related diseases.
503612-47-3 阿派沙班 Apixaban VTE prophylaxis: hip/knee replacement
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